Active Pharmaceutical Ingredient

Naltrexone API Manufacturer & Supplier

CAS: 16590-41-3 Active Pharmaceutical Ingredient IP / BP / EP / USP GMP Certified Aurangabad, Maharashtra, India
Naltrexone API Manufacturer & Supplier — Mediocon Inc
Naltrexone API Manufacturer & Supplier

Product Overview

CAS No: 16590-41-3 | Grade: IP / BP / EP / USP | Category: Active Pharmaceutical Ingredient

Naltrexone API Manufacturer & Supplier

MEDIOCON INC is a trusted global manufacturer and supplier of Naltrexone API, offering premium-quality pharmaceutical-grade active pharmaceutical ingredients for pharmaceutical manufacturing, formulation development, analytical testing, quality control, stability studies, and research applications. Every batch is manufactured under stringent quality management systems to ensure exceptional purity, consistency, and compliance with international pharmaceutical standards.

Naltrexone is a potent opioid receptor antagonist widely used in pharmaceutical formulations for the management of opioid dependence and alcohol use disorder. It works by competitively blocking opioid receptors, preventing the euphoric and sedative effects of opioid drugs while helping reduce alcohol cravings. Naltrexone is also investigated in low-dose formulations (LDN) for autoimmune diseases, chronic pain syndromes, inflammatory disorders, and neurological research. Owing to its well-established pharmacological profile, Naltrexone is extensively utilized in pharmaceutical research, formulation development, analytical method validation, process optimization, stability studies, and quality assurance programs.

MEDIOCON INC supplies premium-quality Naltrexone API to pharmaceutical manufacturers, formulation companies, contract research organizations (CROs), contract development and manufacturing organizations (CDMOs), universities, research institutes, and analytical laboratories worldwide. Comprehensive documentation including Certificate of Analysis (COA), Material Safety Data Sheet (MSDS), Technical Data Sheet (TDS), and regulatory support documents is available upon request.

Product Specifications

Product NameNaltrexone API Manufacturer & Supplier
CAS Number16590-41-3
CategoryActive Pharmaceutical Ingredient
GradeIP / BP / EP / USP
AppearanceWhite to Off-White Crystalline Powder
StandardsIP / BP / EP / USP Compliant

Analytical Specifications

ParameterSpecification
AppearanceWhite to Off-White Crystalline Powder
IdentificationIR, UV & HPLC Compliant
Assay (HPLC)98.0% – 102.0%
Loss on DryingNMT 0.50%
Residue on IgnitionNMT 0.10%
Heavy MetalsNMT 10 ppm
pH (1% Solution)4.5 – 6.5
Individual ImpurityNMT 0.50%
Total ImpuritiesNMT 1.00%
Water ContentNMT 0.50%
Melting Point168°C – 172°C
SolubilityFreely soluble in methanol; slightly soluble in water and ethanol

Sourcing, Regulatory & Export Information

Mediocon Inc is a GMP-certified API manufacturer and bulk pharmaceutical ingredient supplier based in Aurangabad, Maharashtra, India. We specialise in supplying Naltrexone API Manufacturer & Supplier (CAS 16590-41-3) and over 1,000 other Active Pharmaceutical Ingredients, excipients, herbal extracts, and nutraceutical ingredients to pharmaceutical manufacturers worldwide.

Our Naltrexone API Manufacturer & Supplier is manufactured under strict quality management protocols compliant with WHO-GMP, ISO 9001:2015, and major pharmacopoeial standards (IP, BP, USP, EP). Every batch undergoes full analytical testing before release with a Certificate of Analysis.

Export Markets

  • USA — FDA-registered facility; DMF support available for ANDA/NDA filings
  • Europe — EMA-compliant documentation; CEP/EDMF support on request
  • Africa & Middle East — WHO-GMP certified; competitive pricing for emerging markets
  • Southeast Asia — established logistics network; temperature-controlled shipments
  • India domestic — schedule H/X compliance; all state licensing documentation provided

Quality & Compliance

  • ISO 9001:2015 certified quality management system
  • GMP-certified manufacturing facility, Aurangabad, Maharashtra
  • Full batch traceability from raw material to finished API
  • Dedicated QA team for customer audits and regulatory queries

Frequently Asked Questions — Naltrexone API Manufacturer & Supplier

What is Naltrexone API?
Naltrexone API is an opioid receptor antagonist used in pharmaceutical formulations for the treatment of opioid dependence and alcohol use disorder.
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