Active Pharmaceutical Ingredient

Ruboxistaurin — CAS 169939-94-0 API Manufacturer & Supplier in India

Also known as: LY-333531; Arxxant

GMP Certified IP / BP / EP / USP Protein Kinase C Beta Inhibitor Aurangabad, India
Ruboxistaurin API Supplier Manufacturer Aurangabad Maharashtra India — Mediocon Inc
Ruboxistaurin IP / BP / EP / USP  |  GMP Certified  |  Mediocon Inc, Maharashtra, India
CAS No: 169939-94-0

Product Overview

Ruboxistaurin is a high-purity Active Pharmaceutical Ingredient (API) classified under Protein Kinase C Beta Inhibitor. Mediocon Inc manufactures GMP-compliant Ruboxistaurin at its state-of-the-art facility in Aurangabad, Maharashtra, India, supplying pharmaceutical companies worldwide with consistent quality and full regulatory documentation.

Therapeutic Applications
  • Diabetic retinopathy
  • Diabetic macular oedema
  • PKCβ-mediated vascular complications in diabetes
  • Peripheral neuropathy associated with diabetes

Technical Specifications

ParameterSpecification
CAS Number169939-94-0
Molecular FormulaC₂₈H₂₉N₅O₂
Molecular Weight483.57 g/mol
GradeIP / BP / EP / USP
CategoryProtein Kinase C Beta Inhibitor
AssayNLT 98.0%
Loss on DryingNMT 0.5%
Heavy MetalsNMT 20 ppm
Residue on IgnitionNMT 0.1%
Microbial LimitsComplies with pharmacopoeia
IdentificationIR, HPLC Compliant
Batch NoRUB/24032026
Mfg DateMAR 2026
Exp DateFEB 2031
Packing25 kg HDPE drums / as per requirement

Quality & Compliance

  • GMP Certified manufacturing facility in Aurangabad, Maharashtra, India
  • Full pharmacopoeial compliance: IP / BP / EP / USP standards
  • Complete documentation: Certificate of Analysis (CoA), MSDS, Certificate of Origin
  • Stringent in-process quality control at every manufacturing stage
  • HPLC purity testing and spectroscopic identification (IR, NMR)
  • Cold-chain and controlled-environment storage facilities available
  • Exported to 40+ countries with full regulatory support
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