Levocabastine API is a synthetic, highly selective histamine H1-receptor antagonist belonging to the piperidine derivative class of antihistamines. It is a stereochemically defined antihistaminic compound developed for the management of histamine-mediated allergic symptoms. Levocabastine acts primarily on peripheral H1 receptors, thereby reducing the physiological effects of histamine that contribute to allergic manifestations such as itching, redness, sneezing and watery discharge.
Chemically, Levocabastine is identified as 1-[4-cyano-4-(4-fluorophenyl)piperidin-3-yl]-N-(4-methylphenyl)piperidine-4-carboxamide. It has the molecular formula C₂₆H₂₉FN₄O, molecular weight approximately 416.54 g/mol, and CAS number 79547-94-9.
Levocabastine has been particularly associated with topical ophthalmic and nasal pharmaceutical formulations, where its selective H1-antagonist activity is used for the symptomatic management of allergic conjunctivitis and allergic rhinitis. Its peripheral antihistaminic activity makes it relevant to pharmaceutical development involving localized allergy treatment.
MEDIOCON INC supplies Levocabastine for applicable pharmaceutical manufacturing, formulation development, analytical research, quality-control testing and bulk API requirements, subject to product availability, applicable regulatory requirements and batch-specific documentation.
| Parameter | Specification |
|---|---|
| Appearance | White to off-white crystalline powder |
Mediocon Inc is a GMP-certified API manufacturer and bulk pharmaceutical ingredient supplier based in Aurangabad, Maharashtra, India. We specialise in supplying Levocabastine API Manufacturer & Supplier in India | MEDIOCON INC (CAS 79547-94-9) and over 1,000 other Active Pharmaceutical Ingredients, excipients, herbal extracts, and nutraceutical ingredients to pharmaceutical manufacturers worldwide.
Our Levocabastine API Manufacturer & Supplier in India | MEDIOCON INC is manufactured under strict quality management protocols compliant with WHO-GMP, ISO 9001:2015, and major pharmacopoeial standards (IP, BP, USP, EP). Every batch undergoes full analytical testing before release with a Certificate of Analysis.
Export Markets
Quality & Compliance